U-69,593

U-69,593
Clinical data

ATC code	none
Identifiers
IUPAC name N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl)-1-oxaspiro[4.5]dec-8-yl]acetamide
CAS Number	96744-75-1
PubChem CID	105104
IUPHAR/BPS	1655
ChemSpider	94828
ChEBI	CHEBI:73357^Y
ChEMBL	CHEMBL440765
Chemical and physical data
Formula	C₂₂H₃₂N₂O₂
Molar mass	356.50 g/mol
3D model (Jmol)	Interactive image
SMILES O=C(N([C@H]3CC[C@]1(OCCC1)C[C@@H]3N2CCCC2)C)Cc4ccccc4

U-69,593 is a drug which acts as a potent and selective κ₁-opioid receptor agonist. In animal studies it has been shown to produce antinociception,anti-inflammation,anxiolysis (at low doses),respiratory depression, and , while having little effect on gastrointestinal motility. It also inhibits the peripheral, though not central secretion of and vasopressin in rats.

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Wikipedia

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